Mette Rosenkilde
Professor
- 2011
- Published
Allosteric and orthosteric sites in CC chemokine receptor (CCR5), a chimeric receptor approach
Thiele, S., Steen, A., Jensen, P. C., Mokrosinski, J., Frimurer, Thomas Michael & Rosenkilde, Mette, 2011, In: Journal of Biological Chemistry. 286, 43, p. 37543-54 12 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
EBI2, GPR18 and GPR17--three structurally related, but biologically distinct 7TM receptors
Nørregaard, K., Benned-Jensen, T. & Rosenkilde, Mette, 2011, In: Current Topics in Medicinal Chemistry. 11, 6, p. 618-28 11 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Homozygous carriers of the G allele of rs4664447 of the glucagon gene (GCG) are characterised by decreased fasting and stimulated levels of insulin, glucagon and glucagon-like peptide (GLP)-1
Torekov, S. S., Ma, L., Grarup, N., Hartmann, B., Hainerová, I. A., Kielgast, U., Kissow, H., Rosenkilde, M., Lebl, J., Witte, D. R., Jørgensen, T., Sandbaek, A., Lauritzen, T., Madsen, O. D., Wang, J., Linneberg, A., Madsbad, S., Holst, J. J., Hansen, T., Pedersen, O. & 1 others, , 2011, In: Diabetologia. 54, 11, p. 2820-31 12 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Reversed binding of a small molecule ligand in homologous chemokine receptors – differential role of extracellular loop 2.
Rummel, P. C., Thiele, S., Steen, A. M. F., Elder, A., Kolbech, R., Ghosh, S., Frimurer, Thomas Michael & Rosenkilde, Mette, 2011, In: British Journal of Pharmacology. 166Research output: Contribution to journal › Journal article › Research › peer-review
- Published
The E92K melanocortin 1 receptor mutant induces cAMP production and arrestin recruitment but not ERK activity indicating biased constitutive signaling
Benned-Jensen, T., Mokrosinski, J. & Rosenkilde, Mette, 2011, In: P L o S One. 6, 9, p. e24644Research output: Contribution to journal › Journal article › Research › peer-review
- 2010
- Published
Treatment of insulin resistance and obesity by stimulating GLP-1 release
Hansen, Harald S., Diep, T. A., Holst, Jens Juul, Rosenkilde, Mette & Andersen, N. W., 29 Dec 2010, IPC No. A61K 31/23, Patent No. PCT/DK2010/050161, 24 Jun 2010Research output: Patent
- Published
Distinct expression and ligand-binding profiles of two constitutively active GPR17 splice variants
Benned-Jensen, T. & Rosenkilde, Mette, Mar 2010, In: British Journal of Pharmacology. 159, 5, p. 1092-105 14 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Targeting CXCR4 in HIV Cell-Entry Inhibition
Steen, A., Schwartz, Thue W. & Rosenkilde, Mette, 2010, In: Mini reviews in medicinal chemistry. 9, 14, p. 1605-21 16 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
The minor binding pocket: a major player in 7TM receptor activation
Rosenkilde, Mette, Benned-Jensen, T., Frimurer, T. M. & Schwartz, Thue W., 2010, In: Trends in Pharmacological Sciences. 31, 12, p. 567-574 8 p.Research output: Contribution to journal › Journal article › Research › peer-review
- 2009
- Published
The role of transmembrane segment II in 7TM receptor activation
Benned-Jensen, T. & Rosenkilde, Mette, Jun 2009, In: Current Molecular Pharmacology. 2, 2, p. 140-8 9 p.Research output: Contribution to journal › Journal article › Research › peer-review
ID: 3361
Most downloads
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762
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Pharmacokinetics of oral and intravenous melatonin in healthy volunteers
Research output: Contribution to journal › Journal article › Research › peer-review
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440
downloads
Differential CCR7 Targeting in Dendritic Cells by Three Naturally Occurring CC-Chemokines
Research output: Contribution to journal › Journal article › Research › peer-review
Published -
372
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Biased signaling of lipids and allosteric actions of synthetic molecules for GPR119
Research output: Contribution to journal › Journal article › Research › peer-review
Published