Research areas

  1. Published

    Factors that restrict the intestinal cell permeation of cyclic prodrugs of an opioid peptide (DADLE): Part I. Role of efflux transporters in the intestinal mucosa

    Ouyang, H., Chen, W., Andersen, T. E., Steffansen, B. & Borchardt, R. T., 2009, In: Journal of Pharmaceutical Sciences. 98, 1, p. 337-348

    Research output: Contribution to journalJournal articleResearchpeer-review

  2. Published

    Fast prediction of cytochrome P450 mediated drug metabolism

    Rydberg, P. Å. A., Poongavanam, V., Oostenbrink, C. & Olsen, L., 2009, In: ChemMedChem. 4, 12, p. 2070-2079

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Published

    Fate and antibacterial potency of anticoccidal drugs and their main abiotic degradation products

    Hansen, M., Krogh, K. A., Brandt, A., Christensen, Jan H. & Halling-Sørensen, B., 2009, In: Environmental Pollution. 157, 2, p. 474-480 7 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    Fishing for contaminants in McMurdo sound: Antarctica: Analytical methods

    Ghosh, R., Hageman, K., Björklund, B. E., Lamare, M., Metcalf, V. & Lokman, M., 2009.

    Research output: Contribution to conferencePosterCommissioned

  5. Published

    Formation mechanism of insulin fibrils and structural aspects of the insulin fibrillation process

    Jensen, M. G., Frøkjær, Sven & Vestergaard, Bente, 2009, In: Current Protein and Peptide Science. 10, 5, p. 509-528

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Published

    Frequent amplifications and deletions of G1/S-phase trasition genes, CCND1 and MYC in early breast cancers: a potential role in G1/S escape

    Jensen, L. B., Bartlett, J. M. S., Witton, C. J., Kirkegaard, T., Brown, S., Müller, S., Campbell, C., Cooke, T. G. & Nielsen, K. V., 2009, In: Cancer Biomarkers. 5, 1, p. 41-49

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    Full domain closure of the ligand-binding core of the ionotropic glutamate receptor iGluR5 induced by the high affinity agonist dysiherbaine and the functional antagonist 8,9-dideoxyneodysiherbaine

    Frydenvang, Karla Andrea, Lash, L. L., Naur, P., Postila, P. A., Pickering, Darryl S, Smith, C. M., Gajhede, Michael, Sasaki, M., Sakai, R., Pentikäinen, O. T., Swanson, G. T. & Kastrup, Jette Sandholm Jensen, 2009, In: Journal of Biological Chemistry. 284, 21, p. 14219-14229

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published

    Functional characterization of GABA transporters: Emphasis on betaine-GABA transporter 1 and its role in seizure management

    Madsen, K. K., 2009, København: Museum Tusculanum. 54 p.

    Research output: Book/ReportPh.D. thesis

  9. Published

    Functional significance of brain glycogen in sustaining glutamatergic neurotransmission

    Sickmann, H. M., Walls, Anne Byriel, Schousboe, Arne, Bouman, S. D. & Waagepetersen, Helle S., 2009, In: Journal of Neurochemistry. 109, Suppl. 1, p. 80-86 7 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  10. Published

    GABA synthesis from ß-hydroxybutyrate and glucose is differentially affected by neuronal activity in cultured GABAergic neurons

    Lund, Trine Meldgaard, Risa, O., Sonnewald, U., Schousboe, Arne & Waagepetersen, Helle S., 2009, In: Journal of Neurochemistry. s2, p. 95

    Research output: Contribution to journalConference abstract in journalResearch

  11. Published

    GABAA-receptoren: Bedre modeller - bedre lægemidler

    Frølund, Bente, Sander, T., Hansen, H. & Balle, T., 2009, In: Lægemiddelforskning. p. 31-33

    Research output: Contribution to journalJournal articleCommunication

  12. Published

    GABAergic actions on cholinergic laterodorsal tegmental neurons: Implications for control of behavioral state

    Kohlmeier, Kristi Anne & Kristiansen, Uffe, 2009, In: Journal of Neuroscience.

    Research output: Contribution to journalConference abstract in journalResearch

  13. Published

    GAD65 is essential for the maintenance of GABA homeostasis

    Smeland, O., Walls, A. B., Eyolfsson, E. M., Schousboe, Arne, Waagepetersen, Helle S. & Sonnewald, U., 2009, In: Journal of Neurochemistry. p. 51-51

    Research output: Contribution to journalConference abstract in journalResearch

  14. Published

    GAD65 is essential for the maintenance of GABA homeostasis

    Walls, A. B., Eyolfsson, E. M., Sonnewald, U., Vestergaard, H. T., Hansen, S. L., Schousboe, I. E., Schousboe, Arne & Waagepetersen, Helle S., 2009, In: Journal of Neurochemistry. s1, p. 292-292

    Research output: Contribution to journalConference abstract in journalResearch

  15. Published

    Gaboxadol bliver absorberet via en aminosyretransportør

    Broberg, M. L., Holm, R., Jensen, K. G., Larsen, Birger Brodin & Nielsen, C. U., 2009, In: Lægemiddelforskning. p. 22-24

    Research output: Contribution to journalJournal articleCommunication

  16. Published

    Gamma-aminobutyric acid (GABA)

    Schousboe, Arne & Waagepetersen, Helle S., 2009, Encyclopedia of neuroscience. Squire, L. R. (ed.). Academic Press, Vol. 4. p. 511-515

    Research output: Chapter in Book/Report/Conference proceedingEncyclopedia chapterResearch

  17. Published

    Genetic control of disease in an experimental model for Sjögren's syndrome

    Andersson, Åsa, 2009, In: Arthritis Research & Therapy. 11, 1, p. 102

    Research output: Contribution to journalJournal articleResearchpeer-review

  18. Published

    Glial glutamate and GABA metabolism    

    Waagepetersen, Helle S. & Schousboe, Arne, 2009, Encyclopedia of neuroscience. Squire, L. R. (ed.). Academic Press, Vol. 4. p. 789-792

    Research output: Chapter in Book/Report/Conference proceedingEncyclopedia chapterResearch

  19. Published

    Glial modulation of excitability via glutamate and GABA transporters

    Schousboe, Arne & White, H. S., 2009, Encyclopedia of basic epilepsy research. Schwartzkroin, P. A. (ed.). Academic Press, Vol. 1. p. 397-401

    Research output: Chapter in Book/Report/Conference proceedingEncyclopedia chapterResearch

  20. Published

    Glutamate uptake triggers transporter-mediated GABA release from astrocytes

    Héja, L., Barabás, P., Nyitrai, G., Kékesi, K. A., Lasztóczi, B., Toke, O., Tárkányi, G., Madsen, K. K., Schousboe, Arne, Dobolyi, Á., Palkovits, M. & Kardos, J., 2009, In: PLoS ONE. 4, 9, p. e7153-e7153

    Research output: Contribution to journalJournal articleResearchpeer-review

  21. Published

    Glutamatergic neurotransmission under physiological and diabetic conditions - involvement of brain glycogen

    Sickmann, H. M., 2009, København: Det Farmaceutiske Fakultet. 81 p.

    Research output: Book/ReportPh.D. thesis

  22. Published

    Helping hand: patientens forlængede arm

    Christensen, A. & Hansen, E. H., 2009, In: Lægemiddelforskning. p. 40-42

    Research output: Contribution to journalJournal articleCommunication

  23. Published

    Heterocyclic pentafluorophenyl sulfonate esters as shelf stable alternatives to sulfonyl chlorides

    Bornholdt, J., Fjære, K. W., Felding, J. & Kristensen, Jesper Langgaard, 2009, In: Tetrahedron. 65, 45, p. 9280-9284

    Research output: Contribution to journalJournal articleResearchpeer-review

  24. Published

    Histone demethylases

    Clausen, Rasmus Prætorius, Pedersen, M. T. & Helin, K., 2009, Epigenetic targets in drug discovery. Sippl, W. & Jung, M. (eds.). Weinheim: Wiley-VCH, Vol. 42. p. 269-290 (Methods and Principles in Medicinal Chemistry, Vol. 42).

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearch

  25. Published

    Hypoglemic activity of Iraqi Rheum ribes root extract

    Naqishbandi, A. M., Josefsen, K., Pedersen, M. E. & Jäger, A. K., 2009, In: Pharmaceutical Biology. 47, 5, p. 380-383

    Research output: Contribution to journalJournal articleResearchpeer-review

  26. Published

    Identification of reaction products between drug substances and excipients by HPLC-SPE-NMR: Ester and amide formation between citric acid and 5-aminosalicylic acid

    Larsen, J. T., Stærk, Dan, Cornett, Claus, Hansen, S. H. & Jaroszewski, J. W., 2009, In: Journal of Pharmaceutical and Biomedical Analysis. 49, p. 839-842

    Research output: Contribution to journalJournal articleResearchpeer-review

  27. Published

    Impact of adult atopic dermatitis on topical drug penetration: assessment by cutaneous microdialysis and tape stripping

    Garcia Ortiz, P., Hansen, S. H., Shah, V. P., Menné, T. & Benfeldt, E., 2009, In: Acta Dermato Venereologica. 89, 1, p. 33-38 5 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  28. Published

    Impact of carriers in oral absorption: permaeation across Caco-2 cells for the organic anions estrone-3-sulfate and glipizide

    Gram, L. K., Rist, G. M., Lennernäs, H. & Steffansen, B., 2009, In: European Journal of Pharmaceutical Sciences. 37, p. 378-386

    Research output: Contribution to journalJournal articleResearchpeer-review

  29. Published

    Impact of the malate-aspartate shuttle in glutamate neurotransmission

    Waagepetersen, Helle S., Bak, Lasse Kristoffer, Lund, Trine Meldgaard, Walls, A. B., Sonnewald, U. & Schousboe, Arne, 2009, In: Journal of Neurochemistry. s1, p. 9

    Research output: Contribution to journalConference abstract in journalResearch

  30. Published

    Impact of transporters in oral absorption: a case study of in vitro and in vivo organic anion absorption

    Gram, L. K., Rist, G. M. & Steffansen, B., 2009, In: Molecular Pharmaceutics. 6, 5, p. 1457-1465

    Research output: Contribution to journalJournal articleResearchpeer-review

  31. Published

    In situ identification of dimethyl diselenide in hepatocytes treated with methylseleninic acid by membrane inlet mass spectrometry

    Gabel-Jensen, C., Bak, S. A., Lauritsen, F. R., Hansen, H. R., Badolo, L. & Gammelgaard, Bente, 2009, In: Journal of Analytical Atomic Spectrometry. 24, p. 949-952

    Research output: Contribution to journalJournal articleResearchpeer-review

  32. Published

    Increased litter size and super-ovulation rate in congenic C57BL mice carrying a polymorphic fragment of NFR/N origin at the Fecq4 locus of chromosome 9

    Liljander, M., Andersson, Åsa, Holmdahl, R. & Mattsson, R., 2009, In: Genetics Research. 91, 4, p. 259-65 6 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  33. Published

    Increasing process understanding by analyzing complex interactions in experimental data

    Naelapaa, K., Alleso, M., Kristensen, H. G., Bro, Rasmus, Rantanen, Jukka & Bertelsen, P., 2009, In: Journal of Pharmaceutical Sciences. 98, 5, p. 1852-1861

    Research output: Contribution to journalJournal articleResearchpeer-review

  34. Published

    Ind i hjernen med nye stoffer

    Clausen, Rasmus Prætorius, Nielsen, S. D., Kristensen, Jesper Langgaard & Hansen, K. B., 2009, In: Lægemiddelforskning. p. 34-36

    Research output: Contribution to journalJournal articleCommunication

  35. Published

    Influence of the solid form of siramesine hydrochloride on its behaviour in aqueous environments

    Zimmermann, A., Tian, F., Lopez de Diego, H., Ringkjøbing Elema, M., Rantanen, Jukka, Mullertz, Anette & Hovgaard, L., 2009, In: Pharmaceutical Research. 26, 4, p. 846-854

    Research output: Contribution to journalJournal articleResearchpeer-review

  36. Published

    Information about ADRs explored by pharmacovigilance approaches: a qualitative review of studies on antibiotics, SSRIs and NSAIDs

    Aagaard, L. & Hansen, E. H., 2009, In: BMC Clinical Pharmacology. 9, 4, 14 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  37. Published

    Innovativt nanopartikeldesign bag skræddersyede vacciner

    Nordly, P. J., Agger, E. M., Nielsen, Hanne Mørck & Foged, Camilla, 2009, In: Lægemiddelforskning. p. 19-21

    Research output: Contribution to journalJournal articleResearch

  38. Published

    Interactions of antidepressants with serotonin and norepinephrine transporters: Mutational analysis and structure-activity relationship studies

    Andersen, J., 2009, København: Det Farmaceutiske Fakultet. 185 p.

    Research output: Book/ReportPh.D. thesis

  39. Published

    Intestinal gaboxadol absorption via PAT1 (SLC36A1): modified absorption in vivo following co-administration of L-tryptophan

    Larsen, M., Larsen, R., Jensen, K. G., Larsen, Birger Brodin & Nielsen, C. U., 2009, In: British Journal of Pharmacology. 157, p. 1380-1389

    Research output: Contribution to journalJournal articleResearchpeer-review

  40. Published

    Intramyocellular triglyceride content in man, influence of sex, obesity and glycaemic control

    Haugaard, Steen Bendix, Madsbad, Sten, Mu, Huiling & Vaag, Allan, 2009, In: European Journal of Endocrinology. 161, 1, p. 57-64 8 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  41. Published

    Introduction to the topic "drugs and the environment" and outline of the legislation to assess the environmental risk of drugs

    Halling-Sørensen, B., 2009.

    Research output: Contribution to conferenceConference abstract for conferenceCommissioned

  42. Published

    Investigation of a dual CD chiral CE system for separation of glitazone compounds

    Jamali, B., Bjørnsdottir, I., Cornett, Claus & Hansen, S. H., 2009, In: Electrophoresis. 30, 16, p. 2853-2861

    Research output: Contribution to journalJournal articleResearchpeer-review

  43. Published

    Ketogenic diet is antiepileptogenic in pentylenetetrazole kindled mice and decrease levels of N-acylethanolamines in hippocampus

    Hansen, S. L., Nielsen, A. H., Knudsen, K. E., Artmann, A., Kristiansen, Uffe, Hansen, S. H., Hansen, Harald S. & Petersen, G., 2009, In: Neurochemistry International. 54, 3-4, p. 199-204

    Research output: Contribution to journalJournal articleResearchpeer-review

  44. Published

    Knockdown of GDH indicates its potential impact in sustaining glutamate homeostasis and neurotransmission

    Klawonn, A. M., Bolanos, J. P., Waagepetersen, Helle S. & Schousboe, Arne, 2009, In: Journal of Neurochemistry. s2, p. 105

    Research output: Contribution to journalConference abstract in journalResearch

  45. Published

    Knowledge and insight in relation to functional remission in patients with long-term psychotic disorders

    Alenius, M., Hammarlund-Udenaes, M., Hartvig, P. & Lindström, L., 2009, In: Social Psychiatry and Psychiatric Epidemiology. 45, 5, p. 523-529 7 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  46. Published

    Kombination af konserveringsmidler i cremer nedsætter risikoen for allergi

    Lundov, M. D. & Moesby, L., 2009, In: Lægemiddelforskning. p. 13-15

    Research output: Contribution to journalJournal articleCommunication

  47. Published

    LC-ICP-MS and LC-ESI-(MS)n identification of Se-methylselenocysteine and selenomethionine as metabolites of methylseleninic acid in rat hepatocytes

    Gabel-Jensen, C., Jacobsen, J. O., Skonberg, C., Badolo, L. & Gammelgaard, Bente, 2009, In: Journal of Analytical Atomic Spectrometry. 24, p. 69-75

    Research output: Contribution to journalJournal articleResearchpeer-review

  48. Published

    Laegemiddelstyrelsen bør genoverveje tilladelsen til generisk substitution mellem fentanyldepotplastre

    Christrup, Lona Louring, Jensen, N., Jonsson, T., Sjøgren, P. & Steffansen, B., 2009, In: Ugeskrift for læger. 171, 44, p. 3215

    Research output: Contribution to journalComment/debateResearch

  49. Published

    Ligand binding analyses of the putative peptide transporter YjdL from E. coli display a significant selectivity towards dipeptides

    Ernst, H. A., Pham, A., Hald, H., Kastrup, Jette Sandholm Jensen, Rahman, M. & Mirza, Osman Asghar, 2009, In: Biochemical and Biophysical Research Communications. 389, 1, p. 112-116

    Research output: Contribution to journalJournal articleResearchpeer-review

  50. Published

    Lipid based drug delivery systems for proteins: Physical stability of proteins at the oil-water interface

    Jørgensen, Lene, 2009, VDM Verlag Dr. Müller Aktiengesellschaft & C o. KG.

    Research output: Book/ReportBookpeer-review